SCHEMBL7280195

SCHEMBL7280195

N#CNC(=O)/C=C\N1CCCCC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 2/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
MEN1 O00255 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15710798 0.73
SCHEMBL17397278 0.71 NPC1 (0.36) NPC1MAPTLMNAUSP2ALDH1A1
SCHEMBL15710868 0.70
SCHEMBL4125262 0.68 TSHR (0.40) NPC1MAPTLMNAUSP2ALDH1A1
SCHEMBL4784913 0.68
SCHEMBL4125267 0.68 TSHR (0.40) NPC1MAPTLMNAUSP2ALDH1A1
SCHEMBL15349970 0.67 KMT2A (0.57) NPC1MAPTLMNAALDH1A1MEN1
SCHEMBL15349961 0.67 KMT2A (0.57) NPC1MAPTLMNAALDH1A1MEN1
SCHEMBL27677607 0.67
SCHEMBL319864 0.66 ALDH1A1 (0.41) NPC1MAPTLMNAUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0001633-A1 Processes for preparing tri-heterocyclic substituted methanes and their conversion into further intermediates useful in the preparation of pharmacologically active compounds THE WELLCOME FOUNDATION LIMITED (GB) 1979-05-02 EP disclosed