SCHEMBL7280508

SCHEMBL7280508

NC1(C(=O)O)Cc2cc(O)c(O)cc2C1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 6/20 0.42
ALDH1A1 P00352 4/20 0.40
TDP1 Q9NUW8 3/20 0.40
MAPT P10636 2/20 0.40
RECQL P46063 2/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP3A4 P08684 1/20 0.40
THRB P10828 1/20 0.40
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40
CASP1 P29466 1/20 0.40
BLM P54132 1/20 0.40
CASP7 P55210 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NSD2 O96028 1/20 0.39
FYN P06241 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C19 P33261 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5251204 0.83 GRM4 (0.40) GRM4ALDH1A1TDP1KDM4ENSD2
SCHEMBL5246908 0.83 GRM4 (0.40) GRM4ALDH1A1TDP1KDM4ENSD2
SCHEMBL27795991 0.83 GRM4 (0.40) GRM4ALDH1A1TDP1KDM4ENSD2
SCHEMBL7277003 0.79 HSD17B1 (0.42) GRM4ALDH1A1TDP1MAPTKDM4E
SCHEMBL5245248 0.79 IDO1 (0.44) GRM4ALDH1A1TDP1MAPTKDM4E
SCHEMBL7429811 0.78 MAPT (0.40) GRM4ALDH1A1TDP1MAPTRECQL
SCHEMBL122942 0.77 HDAC9 (0.44) GRM4NSD2GRM6
SCHEMBL29476532 0.77 HDAC9 (0.44) GRM4NSD2GRM6
SCHEMBL7271740 0.77 CXCR5 (0.41) GRM4ALDH1A1CASP1
SCHEMBL30758541 0.77 TDP2 (0.41) GRM4MAPTKDM4EHPGDCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766110-A INHIBITS ANGIOTENSIN CONVERTING ENZYME, HYPOTENSIVE AGENTS RYAN JAMES W (US) 1988-08-23 US disclosed
EP-0073143-B1 NOVEL COMPLEX AMIDO AND IMIDO DERIVATIVES OF CARBOXYALKYL PEPTIDES AND THIOETHERS AND ETHERS OF PEPTIDES Ryan, James Walter (US) 1985-11-21 EP disclosed
EP-0048159-A2 Novel carboxyalkyl peptides and thioethers and ethers of peptides as antihypertensive agents UNIVERSITY OF MIAMI (US) 1982-03-24 EP disclosed