SCHEMBL7280656

SCHEMBL7280656

CC(C)(C)OC(=O)COc1ccc(C(=O)NNC(=O)OCc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
CTSK P43235 2/20 0.52
HDAC1 Q13547 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC2 Q92769 1/20 0.48
NCOR2 Q9Y618 1/20 0.48
MAPT P10636 3/20 0.47
KMT2A Q03164 2/20 0.47
POLB P06746 1/20 0.47
CTDSP1 Q9GZU7 1/20 0.47
TP53 P04637 1/20 0.47
PLA2G4B P0C869 1/20 0.47
PTPN1 P18031 1/20 0.45
CASP1 P29466 1/20 0.45
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
PLAU P00749 1/20 0.44
ELANE P08246 1/20 0.44
SYK P43405 1/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7292267 0.86 SMPD1 (0.47) ALDH1A1CTSKHDAC1MAPTKMT2A
SCHEMBL1968491 0.84 KMT2A (0.55) ALDH1A1MAPTKMT2APLA2G4BPTPN1
SCHEMBL8361241 0.84 HDAC1 (0.53) ALDH1A1HDAC1HDAC3HDAC2NCOR2
SCHEMBL8770370 0.84 TP53 (0.68) ALDH1A1MAPTKMT2APOLBTP53
SCHEMBL864308 0.83 HDAC1 (0.61) ALDH1A1CTSKHDAC1HDAC3HDAC2
SCHEMBL12697639 0.80 ALDH1A1 (0.59) ALDH1A1MAPTKMT2APOLBTP53
SCHEMBL7289218 0.79 HDAC1 (0.56) ALDH1A1HDAC1HDAC3HDAC2MAPT
SCHEMBL24899403 0.78 ITGB3 (0.59) ALDH1A1KMT2ACASP1MEN1
SCHEMBL8336016 0.78 ITGB3 (0.59) ALDH1A1CTSKKMT2ACASP1MEN1
SCHEMBL29115912 0.78 ITGB3 (0.67) PTPN1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5981531-A FOR INHIBITING PLATELET AGGREGATION ZENECA LIMITED (GB) 1999-11-09 US disclosed
US-5760057-A ANTICOAGULANTS ZENECA LIMITED (GB) 1998-06-02 US disclosed
EP-0632016-B1 1,2-Diacylated hydrazine derivatives and their use as cell adhesion inhibitors ZENECA LTD (GB) 1997-04-09 EP disclosed
US-5612373-A ANTICOAGULANTS ZENECA LIMITED (GB) 1997-03-18 US disclosed
WO-1995000472-A1 1,2 DIACYLATED HYDRAZINE DERIVATIVES AND THEIR USE AS ALL ADHESION INHIBITORS ZENECA LIMITED (GB) 1995-01-05 WO disclosed
EP-0632016-A1 1,2-Diacylated hydrazine derivatives and their use as cell adhesion inhibitors ZENECA LIMITED (GB) 1995-01-04 EP disclosed