SCHEMBL7280854

SCHEMBL7280854

CCN(CC)CCN(C)C(=O)C[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CPA1 P15085 7/20 0.53
CPA3 P15088 3/20 0.53
CPB1 P15086 1/20 0.53
CPB2 Q96IY4 1/20 0.53
CYP1A2 P05177 1/20 0.50
MME P08473 1/20 0.47
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46
LMNA P02545 1/20 0.45
FOLH1 Q04609 1/20 0.45
ANPEP P15144 1/20 0.45
RNPEP Q9H4A4 1/20 0.45
DNPEP Q9ULA0 1/20 0.45
SLC1A3 P43003 1/20 0.42
SLC1A2 P43004 1/20 0.42
SLC1A1 P43005 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430228 0.90 BCHE (0.44) CPA1CPA3CPB1CPB2CYP1A2
Hydrochloric Acid SCHEMBL10449746 0.86 CPA1 (0.55) CPA1CPA3CPB1CPB2CYP1A2
SCHEMBL7280064 0.85 CPA1 (0.57) CPA1CPA3CPB1CPB2CYP1A2
SCHEMBL7274920 0.81 CPA1 (0.60) CPA1CPA3CPB1CPB2CYP1A2
SCHEMBL7433358 0.81 CPA1 (0.53) CPA1CPA3CPB1CPB2CYP1A2
SCHEMBL38656098 0.80 CYP1A2 (0.59) CPA1CPA3CPB1CPB2CYP1A2
SCHEMBL6343538 0.79 CPA1 (0.66) CPA1CPA3CPB1CPB2CYP1A2
SCHEMBL6343535 0.79 CPA1 (0.66) CPA1CPA3CPB1CPB2CYP1A2
SCHEMBL7302265 0.78 ANPEP (0.49) CPA1CPA3CPB1CPB2CYP1A2
SCHEMBL7299196 0.78 MMP2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258362-A Enzyme inhibitors, amides with oxetane ring ABBOTT LABORATORIES (US) 1993-11-02 US disclosed
WO-1992022313-A1 RENIN INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-12-23 WO disclosed
EP-0416393-A1 Peptidyl difluorodiol renin inhibitors ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
WO-1989010751-A1 FUNCTIONALIZED PEPTIDYL AMINODIOLS AND -TRIOLS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed
EP-0341602-A2 Renin-inhibiting functionalized peptidyl aminodiols and - triols ABBOTT LABORATORIES (US) 1989-11-15 EP disclosed
EP-0307837-A2 Renin-inhibiting peptidyl heterocycles ABBOTT LABORATORIES (US) 1989-03-22 EP disclosed