SCHEMBL7280973

SCHEMBL7280973

COc1ccc(C[C@H](NC(=O)N2CCN(C)CC2)C(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.56
MAPT P10636 1/20 0.55
ITGB1 P05556 1/20 0.55
ITGA4 P13612 1/20 0.55
ITGB7 P26010 1/20 0.55
KMT2A Q03164 2/20 0.52
FPR2 P25090 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
GFER P55789 1/20 0.52
CTSL P07711 1/20 0.51
MMP1 P03956 1/20 0.51
CA2 P00918 1/20 0.50
ITGB3 P05106 1/20 0.50
ITGA2B P08514 1/20 0.50
LDHA P00338 1/20 0.50
GAA P10253 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7278749 0.90 CYP3A4 (0.61) POLBMAPTITGB1ITGA4ITGB7
SCHEMBL6803415 0.87 BLM (0.56) POLBMAPTITGB1ITGA4ITGB7
SCHEMBL27230807 0.86 POLB (0.74) POLBITGB1ITGA4ITGB7KMT2A
SCHEMBL7266885 0.86 POLB (0.74) POLBITGB1ITGA4ITGB7KMT2A
SCHEMBL7295919 0.83 KMT2A (0.57) POLBITGB1ITGA4KMT2AFPR2
SCHEMBL9556460 0.81 ADORA2A (0.58) ITGB1ITGA4ITGB7KMT2AFPR2
SCHEMBL4361126 0.77 ITGB3 (0.64) KMT2AFPR2CA2ITGB3ITGA2B
SCHEMBL8765951 0.77 LDHA (0.63) ITGA4ITGB7KMT2AFPR2CA2
SCHEMBL10663117 0.77 LDHA (0.63) ITGA4ITGB7KMT2AFPR2CA2
SCHEMBL6438360 0.77 ITGB3 (0.64) KMT2AFPR2CA2ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1989010751-A1 FUNCTIONALIZED PEPTIDYL AMINODIOLS AND -TRIOLS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed
EP-0341602-A2 Renin-inhibiting functionalized peptidyl aminodiols and - triols ABBOTT LABORATORIES (US) 1989-11-15 EP disclosed
EP-0307837-A2 Renin-inhibiting peptidyl heterocycles ABBOTT LABORATORIES (US) 1989-03-22 EP disclosed