SCHEMBL7281995

SCHEMBL7281995

CC1Oc2c(cc(Cl)cc2C(=O)O)NC1=O

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.41
PARP1 P09874 5/20 0.39
AKR1C4 P17516 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36
TRPV1 Q8NER1 5/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7288542 0.85 SERPINH1 (0.41) PARP1TRPV1
SCHEMBL7281859 0.83 PARP1 (0.39) PARP1AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL7288322 0.82 HSD17B10 (0.42) DYRK1APARP1HSD17B10
SCHEMBL5671638 0.80 PARP1 (0.44) PARP1TRPV1
SCHEMBL20138195 0.78 PARP1 (0.41) PARP1TRPV1
SCHEMBL20138193 0.78 PARP1 (0.41) PARP1TRPV1
SCHEMBL2351573 0.77 PARP1 (0.51) PARP1TRPV1
SCHEMBL7289440 0.73 HTR3A (0.58) CYP3A4
Hydrochloric Acid SCHEMBL7279269 0.73 HTR3A (0.48) PARP1
SCHEMBL13672063 0.73 PARP1 (0.38) PARP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0313393-B1 Benzoxazine compounds and pharmaceutical use thereof YOSHITOMI PHARMACEUTICAL (JP) 1994-03-16 EP disclosed
US-4892872-A ANTIEMETICS, ANTINAUSEA YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1990-01-09 US disclosed
EP-0313393-A2 Benzoxazine compounds and pharmaceutical use thereof Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-04-26 EP disclosed