SCHEMBL7282148

SCHEMBL7282148

C=CC[C@@H]1C[C@@H](CNC(=O)CCCc2ccc(NC(=O)OC(C)(C)C)cc2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.43
DRD2 P14416 1/20 0.40
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 2/20 0.39
ALOX12 P18054 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NAMPT P43490 1/20 0.39
GLS O94925 1/20 0.38
FAAH O00519 2/20 0.37
MGLL Q99685 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281972 0.97 SIGMAR1 (0.43) SIGMAR1DRD2ALDH1A1MEN1CYP1A2
SCHEMBL7275472 0.93 SIGMAR1 (0.41) SIGMAR1DRD2ALDH1A1MEN1CYP1A2
SCHEMBL7283356 0.90 SIGMAR1 (0.41) SIGMAR1DRD2ALDH1A1MEN1CYP1A2
SCHEMBL7275568 0.89 SIGMAR1 (0.46) SIGMAR1DRD2ALDH1A1CYP3A4NAMPT
SCHEMBL7284620 0.87 SIGMAR1 (0.43) SIGMAR1DRD2ALDH1A1MEN1CYP1A2
SCHEMBL7275906 0.85 SIGMAR1 (0.46) SIGMAR1DRD2CYP3A4MAPTNPSR1
SCHEMBL7276712 0.83 SIGMAR1 (0.48) SIGMAR1MEN1CYP3A4KMT2AMAPT
SCHEMBL7281888 0.83 NPY1R (0.42) SIGMAR1ALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL7273654 0.83 SIGMAR1 (0.44) SIGMAR1DRD2SMN1; SMN2NAMPTFAAH
SCHEMBL7275050 0.83 SIGMAR1 (0.47) SIGMAR1CYP3A4MAPTNPSR1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed