SCHEMBL7275568

SCHEMBL7275568

C=CC[C@@H]1C[C@@H](CNC(=O)CCc2ccc(CNC(=O)OC(C)(C)C)cc2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.46
LTA4H P09960 2/20 0.39
CACNA1G O43497 2/20 0.38
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
NAMPT P43490 1/20 0.37
ALDH1A1 P00352 2/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
CYP3A4 P08684 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281972 0.92 SIGMAR1 (0.43) SIGMAR1LTA4HNAMPTALDH1A1DRD2
SCHEMBL7282148 0.89 SIGMAR1 (0.43) SIGMAR1CA1CA2NAMPTALDH1A1
SCHEMBL7283356 0.88 SIGMAR1 (0.41) SIGMAR1LTA4HALDH1A1DRD2DRD3
SCHEMBL7275906 0.86 SIGMAR1 (0.46) SIGMAR1CACNA1GCA1CA2NAMPT
SCHEMBL7273654 0.85 SIGMAR1 (0.44) SIGMAR1CA1CA2NAMPTDRD2
SCHEMBL7275472 0.85 SIGMAR1 (0.41) SIGMAR1CA1CA2ALDH1A1DRD2
SCHEMBL7276712 0.84 SIGMAR1 (0.48) SIGMAR1CACNA1GCA1CA2CYP3A4
SCHEMBL7304783 0.84 SIGMAR1 (0.39) SIGMAR1ALDH1A1DRD2DRD3CHRNB4
SCHEMBL7275050 0.83 SIGMAR1 (0.47) SIGMAR1CACNA1GCA1CA2NAMPT
SCHEMBL8881851 0.83 SIGMAR1 (0.38) SIGMAR1LTA4HNAMPTDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed