SCHEMBL7282155

SCHEMBL7282155

CCCCNC(=N)c1ccc(N2CCN(c3ccc(CCC(=O)O)cc3)C2=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 5/20 0.53
ITGB3 P05106 7/20 0.46
ITGA2B P08514 7/20 0.46
HDAC1 Q13547 2/20 0.40
HPGD P15428 1/20 0.39
CYP1A2 P05177 1/20 0.39
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
S1PR3 Q99500 2/20 0.37
S1PR2 O95136 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
FFAR1 O14842 1/20 0.37
FFAR4 Q5NUL3 1/20 0.37
EPHX2 P34913 1/20 0.37
NR1H4 Q96RI1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275502 0.90 S1PR1 (0.44) S1PR1ITGB3ITGA2BHDAC1HPGD
SCHEMBL7275936 0.84 ITGB3 (0.52) S1PR1ITGB3ITGA2BHDAC1FFAR1
SCHEMBL7276092 0.80 ITGB3 (0.46) S1PR1ITGB3ITGA2BHDAC1L3MBTL1
SCHEMBL7274080 0.78 ITGB3 (0.74) S1PR1ITGB3ITGA2B
SCHEMBL7274915 0.78 S1PR1 (0.54) S1PR1ITGB3ITGA2BHDAC1S1PR3
SCHEMBL7274246 0.74 S1PR1 (0.52) S1PR1ITGB3ITGA2BHDAC1L3MBTL1
SCHEMBL8417146 0.74 S1PR1 (0.83) S1PR1HDAC1FFAR1FFAR4
Propylamine SCHEMBL8911584 0.74 S1PR1 (0.55) S1PR1ITGB3ITGA2BL3MBTL1FFAR1
SCHEMBL7271946 0.74 ITGB3 (0.63) S1PR1ITGB3ITGA2B
SCHEMBL7284477 0.74 ITGB3 (0.70) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed