SCHEMBL7275502

SCHEMBL7275502

CCCCNC(=N)c1ccc(N2CCN(c3ccc(CCC(=O)OC)cc3)C2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.44
HDAC1 Q13547 2/20 0.39
CYP1A2 P05177 1/20 0.38
MAPT P10636 2/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
POLB P06746 2/20 0.36
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
LMNA P02545 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7282155 0.90 S1PR1 (0.53) S1PR1HDAC1CYP1A2MAPTMAPK1
SCHEMBL7283797 0.85 HDAC1 (0.43) S1PR1HDAC1MAPTHRH3POLB
SCHEMBL7274577 0.84 HDAC1 (0.42) S1PR1HDAC1MAPTHRH3ITGB3
SCHEMBL7281398 0.82 HDAC1 (0.39) S1PR1HDAC1HRH3ITGB3ITGA2B
Hydrochloric Acid SCHEMBL7272547 0.81 ITGB3 (0.53) HDAC1HRH3ITGB3ITGA2B
SCHEMBL8911203 0.80 HDAC1 (0.39) S1PR1HDAC1MAPTHRH3POLB
SCHEMBL7280993 0.80 HDAC1 (0.46) S1PR1HDAC1MAPTHRH3
SCHEMBL7275720 0.80 HDAC1 (0.39) S1PR1HDAC1MAPTHRH3ITGB3
SCHEMBL7272483 0.78 S1PR1 (0.44) S1PR1HDAC1MAPTSMN1; SMN2HRH3
SCHEMBL7280958 0.78 HDAC1 (0.40) S1PR1HDAC1MAPTHRH3ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed