SCHEMBL7283153

SCHEMBL7283153

CC(C)(N)c1ccc(N2CCN(c3ccc(CCC(=O)O)cc3)C2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.50
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
HDAC1 Q13547 5/20 0.44
RXRA P19793 1/20 0.43
RXRB P28702 1/20 0.43
RXRG P48443 1/20 0.43
NR1H4 Q96RI1 3/20 0.42
EPHX2 P34913 1/20 0.42
PPARD Q03181 2/20 0.42
PPARA Q07869 2/20 0.42
FFAR1 O14842 3/20 0.40
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7282165 0.88 S1PR1 (0.48) S1PR1ITGB3ITGA2BHDAC1RXRA
SCHEMBL7280838 0.86 HDAC1 (0.44) S1PR1HDAC1EPHX2PPARDPPARA
SCHEMBL7275491 0.82 S1PR1 (0.52) S1PR1ITGB3ITGA2BHDAC1RXRA
SCHEMBL7275097 0.82 S1PR1 (0.52) S1PR1ITGB3ITGA2BHDAC1RXRA
SCHEMBL7396722 0.80 S1PR1 (0.52) S1PR1ITGB3ITGA2BHDAC1PPARD
SCHEMBL7285127 0.80 S1PR1 (0.50) S1PR1ITGB3ITGA2BHDAC1RXRA
SCHEMBL7273941 0.79 HDAC1 (0.53) S1PR1ITGB3ITGA2BHDAC1RXRA
SCHEMBL7274246 0.79 S1PR1 (0.52) S1PR1ITGB3ITGA2BHDAC1RXRA
Propylamine SCHEMBL8911584 0.79 S1PR1 (0.55) S1PR1ITGB3ITGA2BRXRARXRB
SCHEMBL7274080 0.78 ITGB3 (0.74) S1PR1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed