SCHEMBL7275097

SCHEMBL7275097

NCCc1ccc(N2CCN(c3ccc(CCC(=O)O)cc3)C2=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.52
ITGB3 P05106 1/20 0.50
ITGA2B P08514 1/20 0.50
PPARD Q03181 1/20 0.47
PPARA Q07869 1/20 0.47
FFAR1 O14842 7/20 0.45
RAB9A P51151 2/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
KMT2A Q03164 1/20 0.43
KEAP1 Q14145 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
HDAC1 Q13547 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
FFAR4 Q5NUL3 3/20 0.40
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275491 0.91 S1PR1 (0.52) S1PR1ITGB3ITGA2BPPARDPPARA
SCHEMBL7275091 0.90 S1PR1 (0.45) S1PR1ITGB3ITGA2BPPARDPPARA
SCHEMBL7272781 0.88 S1PR1 (0.46) S1PR1ITGB3ITGA2BRAB9AMEN1
Propylamine SCHEMBL8911584 0.87 S1PR1 (0.55) S1PR1ITGB3ITGA2BPPARDPPARA
SCHEMBL7274314 0.86 ITGB3 (0.48) S1PR1ITGB3ITGA2BPPARDPPARA
SCHEMBL7396722 0.85 S1PR1 (0.52) S1PR1ITGB3ITGA2BPPARDPPARA
SCHEMBL7273999 0.84 S1PR1 (0.44) S1PR1ITGB3ITGA2BPPARDPPARA
SCHEMBL7283243 0.83 HRH3 (0.44) S1PR1ITGB3ITGA2BHDAC1
SCHEMBL7274080 0.83 ITGB3 (0.74) S1PR1ITGB3ITGA2B
SCHEMBL7282165 0.83 S1PR1 (0.48) S1PR1ITGB3ITGA2BPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed