SCHEMBL7284252

SCHEMBL7284252

CCCOc1ccc2c(c1)C(=O)NC2=O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 10/20 0.63
MAOB P27338 10/20 0.63
KMT2A Q03164 4/20 0.54
MEN1 O00255 3/20 0.54
CASP3 P42574 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.49
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MAPT P10636 2/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
RAB9A P51151 1/20 0.49
PIM1 P11309 1/20 0.47
PIM2 Q9P1W9 1/20 0.47
ATM Q13315 1/20 0.46
CHRNA7 P36544 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11518444 0.93 MAOA (0.66) MAOAMAOBKMT2AMEN1L3MBTL1
SCHEMBL11333313 0.89 MAOA (0.61) MAOAMAOBKMT2AMEN1L3MBTL1
SCHEMBL11411139 0.86 MAOA (0.61) MAOAMAOBKMT2AMEN1CASP3
SCHEMBL21543709 0.79 CA12 (0.50) MAOAMAOBKMT2AMEN1L3MBTL1
SCHEMBL5324236 0.79 TGM2 (0.63) MAOAMAOBKMT2AMEN1CASP3
SCHEMBL11579683 0.77 TOP1 (0.57) MAOAMAOBKMT2AMEN1L3MBTL1
SCHEMBL23051433 0.76 MAPT (0.60) KMT2AMEN1L3MBTL1SMN1; SMN2MAPT
SCHEMBL383690 0.76 MAOA (0.59) MAOAMAOBKMT2AMEN1CASP3
Phthalimide SCHEMBL8397522 0.75 PIM1 (0.53) MAOAMAOBKMT2AMEN1CASP3
SCHEMBL29611540 0.75 MAOA (0.81) MAOAMAOBKMT2AMEN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5854275-A Cyclic imide derivatives PFIZER INC. (US) 1998-12-29 US disclosed
US-5326760-A Aminobutanoic acid compounds having metalloprotease inhibiting properties GLAXO, INC. (US) 1994-07-05 US disclosed
US-5252560-A Cyclic imide derivatives, compositions and use GLAXO INC. (US) 1993-10-12 US disclosed
EP-0520573-A1 Cyclic imide derivatives GLAXO INC. (US) 1992-12-30 EP disclosed
US-4144072-A CONTAINING A PHTHALAZINONE AND A PHTHALIMIDE FUJI PHOTO FILM CO., LTD. (JP) 1979-03-13 US disclosed
US-3933507-A LIGHT INSENSITIVE SILVER SALT, POLYMETHINE SENSITIZER AGFA-GEVAERT, A.G. (DT) 1976-01-20 US disclosed