SCHEMBL7284259

SCHEMBL7284259

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCCN(C)CCC(c2ccccc2)c2ccccc2)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.74
ADRA1A P35348 2/20 0.74
MTOR P42345 2/20 0.74
RAB9A P51151 2/20 0.74
SLC6A3 Q01959 2/20 0.74
MLNR O43193 1/20 0.74
NR1I2 O75469 1/20 0.74
CNR1 P21554 1/20 0.74
HRH1 P35367 1/20 0.74
OPRK1 P41145 1/20 0.74
PDE3A Q14432 1/20 0.74
CYP1A2 P05177 5/20 0.70
CYP3A4 P08684 5/20 0.70
CYP2C9 P11712 5/20 0.70
CYP2C19 P33261 5/20 0.70
MAPT P10636 5/20 0.70
LMNA P02545 4/20 0.70
CYP2D6 P10635 4/20 0.70
TSHR P16473 3/20 0.70
TDP1 Q9NUW8 3/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272697 0.98 ADORA3 (0.73) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL7272469 0.95 CYP1A2 (0.78) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL10411083 0.94 ADORA3 (0.66) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL10411081 0.94 ADORA3 (0.66) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL7275429 0.90 CACNA1C (0.70) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL10409941 0.90 CACNA1C (0.69) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL10409943 0.90 CACNA1C (0.69) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL7274431 0.89 CYP1A2 (0.70) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL7275141 0.88 ADORA3 (0.75) ADORA3ADRA1AMTORRAB9ASLC6A3
SCHEMBL7274957 0.88 CYP1A2 (0.70) ADORA3ADRA1AMTORRAB9ASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153016-A2 Asymmetrical diesters of 1,4-dihydro-2,6-dimethyl-pyridine-3,5-dicarboxylic acid RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1985-08-28 EP claimed
US-4772621-A Antihypertensive diphenylpropyl aminopropyl ester of 1,4-dihydro-2,6-dimethyl-pyridine-3,5-dicarboxylic acid RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1988-09-20 US disclosed
US-4705797-A HYPOTENSIVE AGENTS, VASODILATORS RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1987-11-10 US disclosed
EP-0153016-A2 Asymmetrical diesters of 1,4-dihydro-2,6-dimethyl-pyridine-3,5-dicarboxylic acid RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1985-08-28 EP disclosed