SCHEMBL7284532

SCHEMBL7284532

O=C(N[C@@H](Cn1ccnc1)C(=O)O)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.55
CYP26A1 O43174 5/20 0.54
CTSS P25774 1/20 0.54
CTSK P43235 1/20 0.54
CYP19A1 P11511 2/20 0.52
AGTR2 P50052 1/20 0.49
PADI4 Q9UM07 1/20 0.48
TACR1 P25103 1/20 0.48
ITGB3 P05106 3/20 0.47
ITGAV P06756 2/20 0.47
TBXAS1 P24557 1/20 0.47
PPARG P37231 1/20 0.47
PPARA Q07869 1/20 0.47
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
ITGA2B P08514 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204254 0.80 CYP26A1 (0.44) HRH4CYP26A1CTSSCTSKCYP19A1
SCHEMBL204255 0.80 CYP26A1 (0.44) HRH4CYP26A1CTSSCTSKCYP19A1
SCHEMBL305818 0.80 CASP1 (0.48) CTSSCTSKTACR1ITGB3ITGAV
SCHEMBL305819 0.80 CASP1 (0.48) CTSSCTSKTACR1ITGB3ITGAV
SCHEMBL28473741 0.79 SMN1; SMN2 (0.56) HRH4CTSSCTSKCYP19A1CYP11B1
SCHEMBL2397464 0.79 PPARA (0.47) CTSSCTSKTACR1ITGB3ITGAV
SCHEMBL2401482 0.79 PPARA (0.47) CTSSCTSKCYP19A1TACR1ITGB3
SCHEMBL22236504 0.78 CYP26A1 (0.57) HRH4CYP26A1PADI4
SCHEMBL15132766 0.77 SMN1; SMN2 (0.67) HRH4
SCHEMBL9558096 0.76 ITGB3 (0.60) CTSSCTSKTACR1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0509354-B1 Amino acid derivatives HOFFMANN LA ROCHE (CH) 2000-08-23 EP disclosed
US-5393875-A Hypotensive, cardiotonic and antiischemic agents HOFFMANN-LA ROCHE INC. (US) 1995-02-28 US disclosed
EP-0509354-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-10-21 EP disclosed