SCHEMBL7284586

SCHEMBL7284586

NCc1ccc(C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N2CCC(OCC(=O)O)CC2)cc1

nearest known ligand 0.82

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.82
ITGA2B P08514 8/20 0.82
CYP51A1 Q16850 2/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
ACE P12821 1/20 0.43
CCKBR P32239 1/20 0.43
CHRM2 P08172 1/20 0.42
CHRM3 P20309 1/20 0.42
LNPEP Q9UIQ6 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8382276 1.00 ITGB3 (0.82) ITGB3ITGA2BCYP51A1CA1CA2
Lamifiban SCHEMBL4683 0.90 ITGB3 (1.00) ITGB3ITGA2BCYP51A1CA1CA2
Lamifiban SCHEMBL871446 0.90 ITGB3 (1.00) ITGB3ITGA2BCYP51A1CA1CA2
SCHEMBL7283671 0.90 ITGB3 (0.67) ITGB3ITGA2BCYP51A1CA2KMT2A
SCHEMBL8377721 0.90 ITGB3 (0.67) ITGB3ITGA2BCYP51A1CA2KMT2A
SCHEMBL8383693 0.89 ITGB3 (0.80) ITGB3ITGA2BCYP51A1CA1CA2
SCHEMBL8383686 0.89 ITGB3 (0.80) ITGB3ITGA2BCYP51A1CA1CA2
SCHEMBL8383672 0.89 ITGB3 (0.80) ITGB3ITGA2BCYP51A1CA1CA2
SCHEMBL8383680 0.89 ITGB3 (0.80) ITGB3ITGA2BCYP51A1CA1CA2
SCHEMBL8379660 0.88 ITGB3 (0.75) ITGB3ITGA2BCYP51A1CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656348-B1 Aceric acid derivatives as medicaments HOFFMANN LA ROCHE (CH) 2000-05-03 EP disclosed
US-5973188-A Acetic acid derivatives HOFFMANN-LA ROCHE INC. (US) 1999-10-26 US disclosed
EP-0656348-A2 Aceric acid derivatives as medicaments F. HOFFMANN-LA ROCHE AG (CH) 1995-06-07 EP disclosed