SCHEMBL7284684

SCHEMBL7284684

Clc1cccc(Cl)c1NCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
RAD52 P43351 1/20 0.50
KMT2A Q03164 1/20 0.50
P2RX7 Q99572 3/20 0.46
MAPK1 P28482 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C19 P33261 2/20 0.45
ALDH1A1 P00352 2/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
GBA1 P04062 1/20 0.45
PTPN7 P35236 1/20 0.45
DUSP3 P51452 1/20 0.45
PTPN5 P54829 1/20 0.45
PTPN11 Q06124 1/20 0.45
TAAR1 Q96RJ0 1/20 0.45
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11512770 0.83 KMT2A (0.47) POLBRAD52KMT2AMAPK1CYP1A2
SCHEMBL2316630 0.78 HSD17B10 (0.59) KMT2AALDH1A1TSHRHSD17B10THRB
SCHEMBL5914544 0.78 HSD17B10 (0.53) KMT2AP2RX7ALDH1A1TSHRHSD17B10
SCHEMBL19088393 0.77 P2RX7 (0.52) KMT2AP2RX7ALDH1A1HTTAPP
SCHEMBL112756 0.75 HSD17B10 (0.50) POLBKMT2AP2RX7ALDH1A1TSHR
SCHEMBL5608826 0.74 HTT (0.53) POLBRAD52KMT2AP2RX7MAPK1
SCHEMBL11509365 0.74 IDO1 (0.52) POLBRAD52KMT2AALDH1A1HTT
SCHEMBL10546027 0.74 KMT2A (0.50) POLBRAD52KMT2AMAPK1HTT
SCHEMBL11242607 0.74 CYP1A2 (0.48) KMT2ACYP1A2CYP2D6CYP2C19TSHR
SCHEMBL4389670 0.74 KMT2A (0.55) POLBRAD52KMT2APDE5AAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108047068-A A kind of synthetic method of C14H10Cl2NNaO2 impurity B 河南中帅医药科技股份有限公司 2018-05-18 CN disclosed
US-4758563-A 3-alkoxy-2-aminopropyamines, cardiovascular compositions and use MCNEILAB, INC. (US) 1988-07-19 US disclosed
US-4727072-A HYPOTENSIVE AGENTS MCNEILAB, INC. (US) 1988-02-23 US disclosed
EP-0237191-A1 3-alkoxy-2-aminopropylamines useful as cardiovascular agents McNeilab, Inc. (US) 1987-09-16 EP disclosed
US-4256639-A Process for the synthesis of isatin derivatives AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO (IT) 1981-03-17 US disclosed
US-4152452-A N-BENZYLANILINE AND DERIVATIVES WILLIAM H. RORER, INC. (US) 1979-05-01 US disclosed