SCHEMBL7285129

SCHEMBL7285129

CC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@H](C(=O)N[C@@H](C)C(=O)NC(CC(=O)OC(C)(C)C)C(O)CCCc1ccccc1)C(C)C

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
REN P00797 9/20 0.54
BACE1 P56817 5/20 0.53
BACE2 Q9Y5Z0 3/20 0.53
CASP1 P29466 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275856 0.86 CASP1 (0.49) RENBACE1BACE2CASP1
SCHEMBL7275894 0.86 BACE1 (0.50) RENBACE1BACE2CASP1
SCHEMBL7287204 0.86 CASP1 (0.49) RENBACE1BACE2CASP1
SCHEMBL7284988 0.86 CASP1 (0.49) RENBACE1BACE2CASP1
SCHEMBL30008729 0.79 CASP1 (0.59) RENBACE1BACE2CASP1
SCHEMBL7277216 0.77 BACE1 (0.58) RENBACE1BACE2CASP1
SCHEMBL7277693 0.76 BACE1 (0.58) RENBACE1BACE2CASP1
SCHEMBL7285134 0.76 BACE1 (0.59) RENBACE1BACE2CASP1
SCHEMBL5689425 0.76 CASP1 (0.49) RENBACE1BACE2CASP1
SCHEMBL7747439 0.76 BACE1 (0.57) RENBACE1BACE2CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519748-B1 Peptidyl derivatives as inhibitors of interleukin-1B converting enzyme MERCK & CO INC (US) 1998-09-02 EP disclosed
US-5434248-A Peptidyl derivatives as inhibitors of interleukin-1β converting enzyme MERCK & CO., INC. (US) 1995-07-18 US disclosed
EP-0519748-A2 Peptidyl derivatives as inhibitors of interleukin-1B converting enzyme MERCK & CO. INC. (US) 1992-12-23 EP disclosed