SCHEMBL7285541

SCHEMBL7285541

NCCCCc1cncnc1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 11/20 0.57
CYP2A6 P11509 1/20 0.50
MAOA P21397 1/20 0.48
HRH3 Q9Y5N1 4/20 0.45
HRH4 Q9H3N8 3/20 0.45
HRH2 P25021 2/20 0.44
CHRNA7 P36544 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3529110 0.98 HRH1 (0.60) HRH1CYP2A6MAOAHRH3HRH4
SCHEMBL10423050 0.93 CYP2A6 (0.57) HRH1CYP2A6MAOAHRH3HRH4
Hydrochloric Acid SCHEMBL18985043 0.91 CYP2A6 (0.55) HRH1CYP2A6MAOAHRH3HRH4
SCHEMBL8817088 0.82
SCHEMBL28266356 0.78 CHRNB2 (0.38) HRH1CYP2A6CHRNA7
SCHEMBL10768464 0.76 TDP1 (0.35) HRH1CYP2A6
SCHEMBL4177303 0.76 TDP1 (0.59)
SCHEMBL10350035 0.76 CA2 (0.38) HRH1
SCHEMBL13662376 0.76 ATM (0.35) CYP2A6HRH3HRH4CHRNA7
SCHEMBL15545209 0.74 TDP1 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081131-A Omega-((hetero)alkyl)benz(cd)-indol-2-amines AMERICAN CYANAMID COMPANY (US) 1992-01-14 US disclosed
EP-0094080-B1 PYRIDO(2,1-B)QUINAZOLINE DERIVATIVES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1987-09-09 EP disclosed
EP-0230035-A2 Omega-[(hetero)alkyl]benz[cd]indol-2-amines AMERICAN CYANAMID COMPANY (US) 1987-07-29 EP disclosed
US-4551460-A ANTICOAGULANTS, CARDIOVASCULAR DISORDERS HOFFMANN-LA ROCHE INC. (US) 1985-11-05 US disclosed
EP-0094080-A2 Pyrido(2,1-b)quinazoline derivatives F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-11-16 EP disclosed