SCHEMBL7287147

SCHEMBL7287147

O=C(O)C(CCCOC1CCCCO1)Cc1cccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 10/20 0.47
CYP3A4 P08684 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
KDM4E B2RXH2 2/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD1 P21728 1/20 0.47
SLC6A4 P31645 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47
KCNH2 Q12809 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
KDM4C Q9H3R0 1/20 0.43
KCNA5 P22460 1/20 0.41
SCN5A Q14524 1/20 0.41
FOLH1 Q04609 2/20 0.38
CTNNB1 P35222 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7287152 1.00 HTR2A (0.47) HTR2ACYP3A4MEN1KMT2AKDM4E
SCHEMBL27516798 0.77 KDM4C (0.60) MEN1KMT2ASLC6A4KDM4CKCNA5
SCHEMBL7353938 0.76 CTNNB1 (0.48) MEN1KMT2AFOLH1CTNNB1
SCHEMBL9556717 0.76 CTNNB1 (0.48) MEN1KMT2AFOLH1CTNNB1
SCHEMBL10420794 0.75 CTNNB1 (0.47) HTR2ACYP3A4MEN1KMT2AKDM4E
SCHEMBL28664006 0.74 MEN1 (0.44) HTR2ACYP3A4MEN1KMT2ASLC6A4
SCHEMBL11100163 0.74 HTR2A (0.66) HTR2ACYP3A4MEN1KMT2AKDM4E
SCHEMBL4755681 0.74 HTR2A (0.66) HTR2ACYP3A4MEN1KMT2AKDM4E
SCHEMBL31120330 0.73 KCNA5 (0.58) HTR2ACYP3A4MEN1KMT2AKDM4E
SCHEMBL7280245 0.73 CTNNB1 (0.52) KMT2ACYP1A2FOLH1CTNNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5506356-A RENIN INHIBITORS; HYPOTENSIVE AGENTS BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-04-09 US disclosed
US-5481036-A RENIN INHIBITORS, HYPOTENSIVE AGENTS BANYU PHARMACEUTICAL CO., LTD. (JP) 1996-01-02 US disclosed
US-5319082-A N-acylamino acid derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-06-07 US disclosed
US-5240924-A Dipeptide hypotensives BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-08-31 US disclosed
US-5122523-A Hypotensive agents BANYU PHARMACEUTICAL CO., LTD. (JP) 1992-06-16 US disclosed
EP-0309766-A2 N-acylamino acid derivatives and their use BANYU PHARMACEUTICAL CO., LTD. (JP) 1989-04-05 EP disclosed