SCHEMBL7287307

SCHEMBL7287307

O=S(=O)(Oc1ccc2cnccc2c1)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
HSD11B1 P28845 1/20 0.42
PRKCZ Q05513 1/20 0.40
CYP3A4 P08684 3/20 0.40
IMPDH2 P12268 1/20 0.39
PTGS1 P23219 5/20 0.39
PTGS2 P35354 5/20 0.39
ROCK1 Q13464 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
IKBKB O14920 1/20 0.38
CA9 Q16790 1/20 0.38
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
SLC22A12 Q96S37 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1401395 0.95 CA1 (0.44) CA1CA2HSD11B1PRKCZPTGS1
SCHEMBL9250996 0.85 MAPT (0.38) CA1CA2PRKCZCYP3A4ROCK1
SCHEMBL4056753 0.84 CA1 (0.51) CA1CA2HSD11B1CA9HTR1A
SCHEMBL16863083 0.83 CA1 (0.47) CA1CA2HSD11B1CA9HTR1A
SCHEMBL9250998 0.82 PRKCZ (0.37) CA1CA2PRKCZCYP3A4ROCK1
SCHEMBL13933202 0.81 CA1 (0.49) CA1CA2HSD11B1CA9HTR1A
SCHEMBL598333 0.81 CA1 (0.50) CA1CA2HSD11B1CA9HTR1A
SCHEMBL2422700 0.78 CA1 (0.38) CA1CA2PTGS1PTGS2IKBKB
SCHEMBL1713420 0.78 CA1 (0.61) CA1CA2HSD11B1CA9HTR1A
SCHEMBL29839512 0.78 CA1 (0.61) CA1CA2HSD11B1CA9HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed