SCHEMBL7288917

SCHEMBL7288917

Cc1ccc([C@H]2CC3CC[C@H]([C@@H]2C(=O)O)N3C)cc1

nearest known ligand 0.80

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.74
SLC6A2 P23975 5/20 0.74
SLC6A4 P31645 3/20 0.74
CHRNA1 P02708 1/20 0.71
CHRNG P07510 1/20 0.71
ITGA5 P08648 1/20 0.71
CHRNB1 P11230 1/20 0.71
CHRNB2 P17787 1/20 0.71
CHRNB4 P30926 1/20 0.71
CHRNA3 P32297 1/20 0.71
CHRNA4 P43681 1/20 0.71
CHRND Q07001 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5000882 1.00 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL7288922 1.00 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL5000883 1.00 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL9405507 0.89 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL9405545 0.89 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL9405509 0.89 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL15516162 0.89 SLC6A3 (0.76) SLC6A3SLC6A2SLC6A4
SCHEMBL7088802 0.89 SLC6A3 (0.76) SLC6A3SLC6A2SLC6A4
SCHEMBL7669406 0.89 SLC6A3 (0.76) SLC6A3SLC6A2SLC6A4
SCHEMBL7289188 0.88 SLC6A3 (0.75) SLC6A3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604352-B1 Aryl-substituted heterocyclic compounds NEUROSEARCH AS (DK) 2002-10-09 EP disclosed
EP-0604355-B1 Akyl Substituted heterocyclic compounds NEUROSEARCH AS (DK) 2000-08-09 EP disclosed
US-5554626-A TREATMENT OF PARKINSON*S DISEASE, DRUG ABUSE/DEPENDENCE; COANIE/AMPHETAMINE ADDICTION NEUROSEARCH A/S (DK) 1996-09-10 US disclosed
US-5444070-A TREATING A DISEASE OR DISORDER WHICH IS RESPONSIVE TO THE INHIBITION OF DOPAMINE REUPTAKE BY ADMINISTERING A TROPANE DERIVATIVE NEUROSEARCH A/S (DK) 1995-08-22 US disclosed
US-5374636-A Antidrug abuse, antidepressants, antiParkinson activity NEUROSEARCH A/S (DK) 1994-12-20 US disclosed
US-5369113-A Certain 2,3-diphenyl-2-(1,2,4-oxadiazol-5-yl)tropanes useful as dopamide reuptake inhibitors NEUROSEARCH A/S (DK) 1994-11-29 US disclosed
EP-0604355-A2 Akyl Substituted heterocyclic compounds NEUROSEARCH A/S (DK) 1994-06-29 EP disclosed
EP-0604352-A2 Aryl substituted heterocyclic compounds NEUROSEARCH A/S (DK) 1994-06-29 EP disclosed
EP-0604354-A2 Antidepressant and antiparkinsonian compounds NEUROSEARCH A/S (DK) 1994-06-29 EP disclosed