SCHEMBL9405545

SCHEMBL9405545

CC(=O)[C@@H]1C2CCC(C[C@@H]1c1ccc(C)cc1)N2C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.74
SLC6A2 P23975 5/20 0.74
SLC6A4 P31645 3/20 0.74
CHRNA1 P02708 1/20 0.71
CHRNG P07510 1/20 0.71
ITGA5 P08648 1/20 0.71
CHRNB1 P11230 1/20 0.71
CHRNB2 P17787 1/20 0.71
CHRNB4 P30926 1/20 0.71
CHRNA3 P32297 1/20 0.71
CHRNA4 P43681 1/20 0.71
CHRND Q07001 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9405507 1.00 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL9405509 1.00 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL5000883 0.89 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL7288917 0.89 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL7288922 0.89 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL5000882 0.89 SLC6A3 (0.74) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL9405574 0.88 SLC6A3 (0.75) SLC6A3SLC6A2SLC6A4
SCHEMBL4996786 0.88 SLC6A3 (0.73) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL4996780 0.88 SLC6A3 (0.73) SLC6A3SLC6A2SLC6A4CHRNA1CHRNG
SCHEMBL9405578 0.88 SLC6A3 (0.75) SLC6A3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5342949-A Decomposing vinyldiazomethnaes in presence of pyrroles to provide bicyclic ring, which is then reacted with aryl Grignard reagent in presence of copper salt WAKE FOREST UNIVERSITY (US) 1994-08-30 US disclosed
US-5262428-A Compounds for treatment of drug dependency WAKE FOREST UNIVERSITY (US) 1993-11-16 US disclosed