SCHEMBL7289002

SCHEMBL7289002

NC(CO)(C(=O)O)c1cccs1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.42
DAO P14920 1/20 0.39
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
NPC1 O15118 3/20 0.37
POLB P06746 2/20 0.37
RAB9A P51151 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HIF1A Q16665 1/20 0.36
ERCC5 P28715 1/20 0.36
FEN1 P39748 1/20 0.36
HPGDS O60760 1/20 0.35
GSK3B P49841 1/20 0.35
CYP1A2 P05177 1/20 0.35
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7289007 1.00 KIF11 (0.42) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL9832653 0.84 KMT2A (0.49) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL5522634 0.84 KMT2A (0.49) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL22445447 0.84 KMT2A (0.49) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL27814402 0.81 HPGD (0.41) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL22394828 0.76 TSHR (0.39) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL10670693 0.76 DAO (0.45) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL599752 0.75 DAO (0.43) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL41617 0.75 DAO (0.43) KIF11DAOCYP2C19KMT2AMEN1
SCHEMBL1421302 0.75 DAO (0.43) KIF11DAOCYP2C19KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0372537-A2 Urea derivatives of dipeptides with enzyme-inhibiting properties, process to make them, compositions containing them and their use HOECHST AKTIENGESELLSCHAFT (DE) 1990-06-13 EP claimed
EP-1003751-A1 HYDROXAMIC ACID SUBSTITUTED FUSED HETEROCYCLIC METALLOPROTEINASE INHIBITORS AMGEN INC. (US) 2000-05-31 EP disclosed
WO-1999006410-A1 HYDROXAMIC ACID SUBSTITUTED FUSED HETEROCYCLIC METALLOPROTEINASE INHIBITORS AMGEN INC. (US) 1999-02-11 WO disclosed
US-5116835-A Hypotensive agents HOECHST AKTIENGESELLSCHAFT (DE) 1992-05-26 US disclosed
EP-0372537-A2 Urea derivatives of dipeptides with enzyme-inhibiting properties, process to make them, compositions containing them and their use HOECHST AKTIENGESELLSCHAFT (DE) 1990-06-13 EP disclosed