SCHEMBL7289474

SCHEMBL7289474

CSc1ccc(CCCN)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 6/20 0.50
MAOA P21397 2/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A3 Q01959 1/20 0.48
HTR2A P28223 2/20 0.45
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA9 Q16790 1/20 0.41
TAAR1 Q96RJ0 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2A6 P11509 1/20 0.41
ESR1 P03372 1/20 0.41
CYP19A1 P11511 1/20 0.41
ESR2 Q92731 1/20 0.41
GAA P10253 1/20 0.41
HRH1 P35367 2/20 0.41
AKT2 P31751 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9718107 0.94 MAOA (0.54) SLC6A4MAOASLC6A2SLC6A3HTR2A
SCHEMBL28210024 0.92 MAOA (0.52) SLC6A4MAOASLC6A2SLC6A3HTR2A
SCHEMBL1570452 0.86 TAAR1 (0.56) SLC6A4MAOASLC6A2SLC6A3HTR2A
SCHEMBL3678682 0.81 MAOA (0.62) MAOASLC6A2HTR2ATAAR1CYP1A2
SCHEMBL8641530 0.80 CA2 (0.50) SLC6A4MAOASLC6A2SLC6A3HTR2A
SCHEMBL7297985 0.78 SLC6A4 (0.45) SLC6A4MAOASLC6A2SLC6A3CA12
SCHEMBL81913 0.78 SLC6A4 (0.51) SLC6A4MAOASLC6A2SLC6A3CA2
SCHEMBL7289466 0.78 SLC6A4 (0.46) SLC6A4MAOASLC6A2SLC6A3CA12
SCHEMBL4460695 0.78 SLC6A4 (0.45) SLC6A4MAOASLC6A2SLC6A3CYP1A2
SCHEMBL5542530 0.78 SLC6A4 (0.45) SLC6A4MAOASLC6A2SLC6A3CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0443560-A2 HIV protease inhibitors BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1991-08-28 EP claimed
EP-0443573-A2 HIV protease inhibitors containing derived amino acids BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1991-08-28 EP claimed
WO-2021102332-A1 TGFBETAR2 INHIBITOR-LRRC15 ANTIBODY CONJUGATES AND USES THEREOF SILVERBACK THERAPEUTICS, INC. (US) 2021-05-27 WO disclosed
EP-0443560-A2 HIV protease inhibitors BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1991-08-28 EP disclosed
EP-0443573-A2 HIV protease inhibitors containing derived amino acids BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1991-08-28 EP disclosed