SCHEMBL7290465

SCHEMBL7290465

COC(=O)N[C@H](C(=O)NN(Cc1ccc(OCc2ccccc2)cc1)CC(O)C(Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NC(=O)c1ccc2ccccc2n1)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 2/20 0.46
ABCB1 P08183 2/20 0.46
OPRK1 P41145 2/20 0.46
GHSR Q92847 2/20 0.46
ABCG2 Q9UNQ0 2/20 0.46
UGT1A1 P22309 2/20 0.46
MLNR O43193 1/20 0.46
NR1I2 O75469 1/20 0.46
SLCO2B1 O94956 1/20 0.46
CCKAR P32238 1/20 0.46
SLCO1B3 Q9NPD5 1/20 0.46
SLCO1B1 Q9Y6L6 1/20 0.46
CTSD P07339 6/20 0.45
CYP3A4 P08684 3/20 0.45
ABCC3 O15438 1/20 0.45
ABCC4 O15439 1/20 0.45
CACNA1F O60840 1/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
TACR2 P21452 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7290464 1.00 ABCB11 (0.46) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL6443032 0.94 CTSD (0.49) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL6443031 0.94 CTSD (0.49) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL7290472 0.92 CYP3A4 (0.42) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL7290476 0.92 CYP3A4 (0.42) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL7394497 0.91 CTSD (0.48) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL7394494 0.91 CTSD (0.48) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL7290460 0.88 UGT1A1 (0.46) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL7288898 0.87 CYP3A4 (0.43) ABCB11ABCB1OPRK1GHSRABCG2
SCHEMBL7288903 0.87 CYP3A4 (0.43) ABCB11ABCB1OPRK1GHSRABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604368-A1 Anti retroviral hydrazine derivatives CIBA-GEIGY AG (CH) 1994-06-29 EP disclosed