SCHEMBL7293221

SCHEMBL7293221

FC(F)(F)Oc1ccc2c(c1)[C]CCO2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 5/20 0.37
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
CHRM5 P08912 1/20 0.34
SCN1A P35498 1/20 0.34
SCN4A P35499 1/20 0.34
KCNH2 Q12809 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34
SCN2A Q99250 1/20 0.34
SCN3A Q9NY46 1/20 0.34
SCN8A Q9UQD0 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
BACE1 P56817 2/20 0.33
CTSD P07339 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7289919 0.88 GPR3 (0.37) GPR3PTGS1PTGS2CHRM5SCN1A
SCHEMBL9586832 0.80 RAB9A (0.41) HPGDSMN1; SMN2ALDH1A1RAB9A
SCHEMBL578279 0.80 RAB9A (0.41) HPGDSMN1; SMN2ALDH1A1RAB9A
SCHEMBL7297788 0.76 MAPT (0.38) KCNH2ALDH1A1RAB9A
SCHEMBL9585550 0.73 FABP6 (0.40) HPGDSMN1; SMN2ALDH1A1RAB9A
SCHEMBL577551 0.73 FABP6 (0.40) HPGDSMN1; SMN2ALDH1A1RAB9A
SCHEMBL7301082 0.72 P2RY1 (0.36) GPR3PTGS1PTGS2BACE1CTSD
SCHEMBL7293216 0.70 PTGS1 (0.41) GPR3PTGS1PTGS2CHRM5SCN1A
SCHEMBL30616492 0.70 CTNNB1 (0.41) GPR3PTGS1PTGS2CHRM5CA12
SCHEMBL17384160 0.70 CTNNB1 (0.41) GPR3PTGS1PTGS2CHRM5CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260444-A Cardiovascular, hypotensive WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed
US-5208245-A Hypotensive agents WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-05-04 US disclosed
EP-0460418-A2 Novel Dihydropyridine derivative WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1991-12-11 EP disclosed