SCHEMBL7294476

SCHEMBL7294476

COC(=O)c1c(OC)n(C2CCN(CCNS(C)(=O)=O)CC2)c2ccc(F)cc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.52
NPSR1 Q6W5P4 3/20 0.52
PMP22 Q01453 2/20 0.52
MEN1 O00255 2/20 0.52
CYP3A4 P08684 2/20 0.52
KMT2A Q03164 2/20 0.52
LMNA P02545 1/20 0.52
PLD2 O14939 10/20 0.43
PLD1 Q13393 9/20 0.43
HTR4 Q13639 3/20 0.42
CYP1A2 P05177 1/20 0.42
ALOX15 P16050 1/20 0.42
NFKB1 P19838 1/20 0.42
GSK3B P49841 1/20 0.40
ALDH1A1 P00352 2/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
DRD2 P14416 1/20 0.39
HTR3A P46098 2/20 0.38
GLA P06280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294480 0.85 CYP2C9 (0.55) CYP2C9NPSR1PMP22MEN1CYP3A4
SCHEMBL16504002 0.82 CYP2C9 (0.66) CYP2C9NPSR1PMP22MEN1CYP3A4
SCHEMBL7358517 0.80 CYP2C9 (0.49) CYP2C9NPSR1PMP22MEN1CYP3A4
SCHEMBL7301907 0.79 CYP2C9 (0.53) CYP2C9NPSR1PMP22MEN1CYP3A4
SCHEMBL7303226 0.75 CYP2C9 (0.49) CYP2C9NPSR1PMP22MEN1CYP3A4
SCHEMBL7358522 0.74 HTR4 (0.60) CYP2C9NPSR1PMP22MEN1CYP3A4
SCHEMBL7300888 0.71 HTR4 (0.77) CYP2C9NPSR1PMP22MEN1CYP3A4
Hydrochloric Acid SCHEMBL7291228 0.71 HTR4 (0.76) CYP2C9NPSR1PMP22MEN1CYP3A4
SCHEMBL29385613 0.71 CYP2C9 (0.94) CYP2C9NPSR1PMP22MEN1CYP3A4
SCHEMBL2940596 0.71 CYP2C9 (0.94) CYP2C9NPSR1PMP22MEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP disclosed
WO-1992014727-A1 3-PIPERIDINYLMETHYLCARBOXYLATE SUBSTITUTED INDOLES GLAXO GROUP LIMITED (GB) 1992-09-03 WO disclosed
EP-0501322-A1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LIMITED (GB) 1992-09-02 EP disclosed