SCHEMBL7358517

SCHEMBL7358517

COC(=O)c1cn(C2CCN(CCNS(C)(=O)=O)CC2)c2ccc(F)cc12

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.49
PMP22 Q01453 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
CYP3A4 P08684 1/20 0.49
KMT2A Q03164 1/20 0.49
HTR4 Q13639 2/20 0.49
CYP1A2 P05177 1/20 0.49
ALOX15 P16050 1/20 0.49
NFKB1 P19838 1/20 0.49
HTR3A P46098 13/20 0.47
ASH1L Q9NR48 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703205 0.90 HTR4 (0.52) CYP2C9PMP22NPSR1MEN1LMNA
SCHEMBL7358522 0.83 HTR4 (0.60) CYP2C9PMP22NPSR1MEN1LMNA
SCHEMBL7294476 0.80 CYP2C9 (0.52) CYP2C9PMP22NPSR1MEN1LMNA
SCHEMBL7300888 0.80 HTR4 (0.77) CYP2C9PMP22NPSR1MEN1LMNA
Hydrochloric Acid SCHEMBL7291228 0.79 HTR4 (0.76) CYP2C9PMP22NPSR1MEN1LMNA
SCHEMBL7305923 0.76 CNR1 (0.50) CYP2C9PMP22NPSR1MEN1LMNA
SCHEMBL7294480 0.75 CYP2C9 (0.55) CYP2C9PMP22NPSR1MEN1LMNA
SCHEMBL9703208 0.74 HTR4 (0.61) CYP2C9PMP22NPSR1MEN1LMNA
SCHEMBL7667532 0.73 HTR3A (0.51) HTR3A
SCHEMBL16504002 0.73 CYP2C9 (0.66) CYP2C9PMP22NPSR1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP disclosed
EP-0501322-A1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LIMITED (GB) 1992-09-02 EP disclosed