SCHEMBL7294608

SCHEMBL7294608

CN=C(N)N1C2CCC1CC(n1cc(C(=O)O)c3ccccc31)C2

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
OPRL1 P41146 1/20 0.47
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
HTR3A P46098 9/20 0.44
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PLK1 P53350 2/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C1 Q04828 1/20 0.34
HTR3E A5X5Y0 2/20 0.34
HTR3B O95264 2/20 0.34
HTR3D Q70Z44 2/20 0.34
HTR3C Q8WXA8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7300839 0.85 KDM4E (0.50) KDM4EOPRM1OPRD1OPRK1OPRL1
SCHEMBL3724624 0.83 HTR3A (0.56) KDM4EOPRM1OPRD1OPRK1OPRL1
SCHEMBL3724622 0.83 HTR3A (0.56) KDM4EOPRM1OPRD1OPRK1OPRL1
SCHEMBL7490360 0.83 HTR3A (0.56) KDM4EOPRM1OPRD1OPRK1OPRL1
SCHEMBL2318444 0.83 HTR3A (0.56) KDM4EOPRM1OPRD1OPRK1OPRL1
Hydrochloric Acid SCHEMBL7296594 0.82 KDM4E (0.50) KDM4EOPRM1OPRD1OPRK1OPRL1
Hydrochloric Acid SCHEMBL467193 0.82 HTR3A (0.55) KDM4EOPRM1OPRD1OPRK1OPRL1
SCHEMBL12486470 0.81 KDM4E (0.69) KDM4EOPRM1OPRD1OPRK1OPRL1
Iodomethane SCHEMBL1309118 0.81 HTR3A (0.54) KDM4EOPRM1OPRD1OPRK1OPRL1
SCHEMBL9582122 0.78 KDM4E (0.46) KDM4EOPRM1OPRD1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5252570-A Amidino and guanidino derivatives B.I. ITALIA (IT) 1993-10-12 US disclosed
EP-0351385-A2 New amidino and guanidino derivatives BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1990-01-17 EP disclosed