SCHEMBL7296629

SCHEMBL7296629

CC(C)(C)OC(=O)[C@@H]1CCCN1C(=O)CNS(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.49
POLB P06746 4/20 0.49
TSHR P16473 3/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 6/20 0.49
ALOX15 P16050 1/20 0.48
MAPT P10636 2/20 0.47
PREP P48147 1/20 0.47
GFER P55789 1/20 0.47
HCRTR1 O43613 1/20 0.46
KMT2A Q03164 1/20 0.46
GAA P10253 2/20 0.45
RECQL P46063 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9225350 0.87 TSHR (0.54) HPGDPOLBTSHRALDH1A1ALOX15
Hydrochloric Acid SCHEMBL7298291 0.86 TSHR (0.53) HPGDPOLBTSHRALDH1A1ALOX15
SCHEMBL8701236 0.83 HPGD (0.55) HPGDPOLBTSHRALDH1A1ALOX15
SCHEMBL7292745 0.79 PREP (0.49) TSHRALDH1A1MAPTPREPKMT2A
SCHEMBL7338507 0.74 ALDH1A1 (0.48) HPGDPOLBTSHRALDH1A1ALOX15
SCHEMBL6786668 0.72 KLK5 (0.46) ALDH1A1MAPTKMT2AGAA
SCHEMBL6786659 0.72 KLK5 (0.46) ALDH1A1MAPTKMT2AGAA
SCHEMBL6783713 0.72 NPC1 (0.48) ALDH1A1KMT2A
SCHEMBL6783707 0.72 NPC1 (0.48) ALDH1A1KMT2A
SCHEMBL13590682 0.72 HPGD (0.64) HPGDPOLBTSHRALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380713-A Serine protease inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-10 US claimed
EP-0526877-A2 Peptide aldehydes as antithrombotic agents Bristol-Myers Squibb Company (US) 1993-02-10 EP claimed
US-5380713-A Serine protease inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-10 US disclosed
EP-0526877-A2 Peptide aldehydes as antithrombotic agents Bristol-Myers Squibb Company (US) 1993-02-10 EP disclosed