SCHEMBL7298232

SCHEMBL7298232

[O]c1cccc(-c2ccc(=O)[nH]n2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.65
LMNA P02545 3/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
PDE4A P27815 3/20 0.51
PDE4B Q07343 3/20 0.51
PDE4C Q08493 3/20 0.51
PDE4D Q08499 3/20 0.51
GPR119 Q8TDV5 2/20 0.49
PDE3B Q13370 5/20 0.49
PDE3A Q14432 5/20 0.49
HPGD P15428 2/20 0.43
TP53 P04637 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10353459 0.89 CYP1A2 (0.74) CYP1A2LMNAKMT2AMEN1PDE4A
SCHEMBL2152938 0.81 CYP1A2 (0.62) CYP1A2LMNAKMT2AMEN1PDE4A
SCHEMBL2829502 0.81 CYP1A2 (0.62) CYP1A2LMNAKMT2AMEN1PDE4A
SCHEMBL4048920 0.81 CYP1A2 (0.62) CYP1A2LMNAKMT2AMEN1PDE4A
SCHEMBL1301730 0.81 CYP1A2 (0.62) CYP1A2LMNAKMT2AMEN1PDE4A
SCHEMBL10066830 0.81 CYP1A2 (0.62) CYP1A2LMNAKMT2AMEN1PDE4A
SCHEMBL11628763 0.81 KMT2A (0.64) CYP1A2LMNAKMT2AMEN1PDE4A
Bromide SCHEMBL11739258 0.79 CYP1A2 (0.61) CYP1A2LMNAKMT2AMEN1PDE4A
Bromide SCHEMBL11742008 0.79 CYP1A2 (0.61) CYP1A2LMNAKMT2AMEN1PDE4A
SCHEMBL482059 0.79 CYP1A2 (1.00) CYP1A2LMNAKMT2AMEN1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed
EP-0400519-A1 2-Hydroxy-n-propylamines, medicaments containing these compounds and method for preparing them Dr. Karl Thomae GmbH (DE) 1990-12-05 EP disclosed