SCHEMBL7298495

SCHEMBL7298495

N#Cc1c(C#N)c(C#N)c2ccccc2c1[O]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
PDE9A O76083 2/20 0.36
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
EGFR P00533 1/20 0.35
SRC P12931 1/20 0.35
MAPK1 P28482 1/20 0.34
STAT3 P40763 1/20 0.34
TSHR P16473 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
HPGD P15428 1/20 0.33
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2546104 0.85 ALDH1A1 (0.59) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL148856 0.80 ALDH1A1 (0.59) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL150623 0.77 ALDH1A1 (0.64) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL29429129 0.77 ALDH1A1 (0.64) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL514645 0.74 ALDH1A1 (0.48) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL5252145 0.73 ALDH1A1 (0.46) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL5252143 0.73 ALDH1A1 (0.46) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL7307452 0.70 CA1 (0.46) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL16213053 0.69 TSHR (0.57) ALDH1A1KDM4EMEN1KMT2AGAA
SCHEMBL4063685 0.69 ALDH1A1 (0.52) ALDH1A1KDM4EMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed