SCHEMBL7298592

SCHEMBL7298592

CCc1cc2c(s1)S(=O)(=O)Cc1cc(=O)n(-c3ccc(Cl)cc3)nc1-2

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.35
MEN1 O00255 4/20 0.34
KMT2A Q03164 4/20 0.34
MAPT P10636 3/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
ALOX12 P18054 1/20 0.33
CHRNA7 P36544 1/20 0.31
KDM4E B2RXH2 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
KCNH2 Q12809 2/20 0.30
OPRK1 P41145 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7377993 0.90 ALDH1A1 (0.36) AOC3MEN1KMT2AMAPTPOLB
SCHEMBL7378334 0.82 LMNA (0.35) AOC3MEN1KMT2AMAPTPOLB
SCHEMBL9396574 0.81 LMNA (0.34) AOC3MEN1KMT2AMAPTPOLB
SCHEMBL7298220 0.79 LMNA (0.36) AOC3MEN1KMT2AMAPTPOLB
SCHEMBL7290031 0.79 ALDH1A1 (0.39) MEN1KMT2AMAPTPOLBGAA
SCHEMBL7289101 0.78 ALDH1A1 (0.40) AOC3MEN1KMT2AMAPTPOLB
SCHEMBL7373573 0.76 AOC3 (0.37) AOC3MEN1KMT2AMAPTPOLB
SCHEMBL7300102 0.76 KMT2A (0.33) AOC3MEN1KMT2AMAPTLMNA
SCHEMBL7297690 0.75 LMNA (0.36) AOC3MEN1KMT2AMAPTPOLB
SCHEMBL10564787 0.75 LMNA (0.45) AOC3MEN1KMT2AMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426018-B1 Thiophene compounds and their pharmaceutical uses YOSHITIOMI PHARMACEUTICAL IND (JP) 1997-08-27 EP disclosed
EP-0729960-A1 Thiophene compounds and their use as intermediates in the preparation of antianxiety drugs, hypnotics, antiepileptic drugs and nuotropics YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-09-04 EP disclosed
US-5329016-A Antianxiety, hypnotic agents, antiepileptic agents or nootropics YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-07-12 US disclosed
US-5175162-A Anxiolytic, antiepilepic agents YOSHITIOMI PHARMACEUTICAL INDUSTRIES LTD. (JP) 1992-12-29 US disclosed
EP-0426018-A2 Thiophene compounds and their pharmaceutical uses YOSHITIOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-05-08 EP disclosed