SCHEMBL7298657

SCHEMBL7298657

NCCOc1cccc(-c2ccc(=O)[nH]n2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
HRH3 Q9Y5N1 7/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
LMNA P02545 2/20 0.44
CHRM2 P08172 1/20 0.42
SLC6A2 P23975 1/20 0.42
ADRA1A P35348 1/20 0.42
HTR3A P46098 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KCNH2 Q12809 1/20 0.42
PDE3B Q13370 2/20 0.42
PDE3A Q14432 2/20 0.42
GSK3B P49841 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10966475 0.86 CYP1A2 (0.50) CYP1A2HRH3GAAMAPTPDE4A
SCHEMBL10967551 0.83 MAPT (0.60) CYP1A2GAAMAPTPDE4APDE4B
SCHEMBL7306800 0.83 HRH3 (0.62) CYP1A2HRH3MAPTPDE4APDE4B
SCHEMBL10969278 0.80 CYP1A2 (0.49) CYP1A2HRH3GAAMAPTPDE4A
SCHEMBL3159466 0.77 CYP1A2 (0.65) CYP1A2MAPTPDE4APDE4BPDE4C
SCHEMBL10353459 0.77 CYP1A2 (0.74) CYP1A2HRH3MAPTPDE4APDE4B
SCHEMBL7296858 0.76 PDE4A (0.56) CYP1A2HRH3MAPTPDE4APDE4B
Bromide SCHEMBL8110043 0.75 HRH3 (0.63) CYP1A2HRH3MAPTPDE4APDE4B
SCHEMBL30745160 0.75 XDH (0.59) CYP1A2MAPTPDE4APDE4BPDE4C
SCHEMBL8791883 0.75 HRH3 (0.63) CYP1A2HRH3MAPTPDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed
EP-0400519-A1 2-Hydroxy-n-propylamines, medicaments containing these compounds and method for preparing them Dr. Karl Thomae GmbH (DE) 1990-12-05 EP disclosed