SCHEMBL7298969

SCHEMBL7298969

CC(C)[C@H](N)C(=O)N[C@@H](Cc1ccccc1)C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)C(C)C

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
BACE1 P56817 1/20 0.50
CTRB1 P17538 3/20 0.49
CA2 P00918 1/20 0.48
LAP3 P28838 2/20 0.46
ANPEP P15144 1/20 0.46
RNPEP Q9H4A4 1/20 0.46
DNPEP Q9ULA0 1/20 0.46
CTSD P07339 1/20 0.46
LMNA P02545 1/20 0.46
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446490 1.00 NPC1 (0.51) NPC1RAB9ABACE1CTRB1CA2
SCHEMBL7332765 0.97 NPC1 (0.51) NPC1RAB9ABACE1CTRB1CA2
SCHEMBL6445202 0.97 NPC1 (0.51) NPC1RAB9ABACE1CTRB1CA2
SCHEMBL6445073 0.97 NPC1 (0.51) NPC1RAB9ABACE1CTRB1CA2
SCHEMBL6444710 0.97 NPC1 (0.51) NPC1RAB9ABACE1CTRB1CA2
Hydrochloric Acid SCHEMBL8536633 0.96 NPC1 (0.50) NPC1RAB9ABACE1CTRB1CA2
Hydrochloric Acid SCHEMBL8535496 0.96 NPC1 (0.50) NPC1RAB9ABACE1CTRB1CA2
SCHEMBL7270703 0.85 CTSD (0.68) CA2CTSD
SCHEMBL7301400 0.84 CA2 (0.56) BACE1CA2CYP3A4MAPK1
SCHEMBL7279585 0.83 CA2 (0.43) NPC1RAB9ABACE1CTRB1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed