SCHEMBL7299583

SCHEMBL7299583

CCOC(=O)C(OC)C1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.46
EED O75530 1/20 0.46
RBBP4 Q09028 1/20 0.46
SUZ12 Q15022 1/20 0.46
EZH2 Q15910 1/20 0.46
AEBP2 Q6ZN18 1/20 0.46
DPP4 P27487 1/20 0.46
RECQL P46063 1/20 0.44
EPHX1 P07099 1/20 0.44
GAA P10253 1/20 0.43
GPR119 Q8TDV5 4/20 0.43
USP2 O75604 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
MMP13 P45452 1/20 0.41
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1873727 0.84 EPHX1 (0.50) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL122218 0.83 GPR119 (0.50) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL27475723 0.82 EPHX1 (0.46) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL17729229 0.82 HPGD (0.47) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL27446359 0.82 DPP4 (0.52) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL5947150 0.82 HPGD (0.47) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL6105487 0.81 HPGD (0.46) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL8328321 0.81 HPGD (0.46) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL6105490 0.81 HPGD (0.46) HPGDEEDRBBP4SUZ12EZH2
SCHEMBL6058985 0.81 GPR119 (0.48) HPGDEEDRBBP4SUZ12EZH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0928793-B1 Thiazole derivatives HOFFMANN LA ROCHE (CH) 2002-05-15 EP disclosed
US-6001855-A REACTING A THIAZOLE DERIVATIVE AND A CYCLIC AMINE DERIVATIVE; INHIBITS BINDING OF ADHESIVE PROTEINS TO THE SURFACE OF DIFFERENT TYPES OF CELL AND ACCORDINGLY INFLUENCE CELL-CELL AND CELL-MATRIX INTERACTIONS HOFFMAN-LA ROCHE INC. (US) 1999-12-14 US disclosed
EP-0928793-A1 Thiazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1999-07-14 EP disclosed