SCHEMBL7299678

SCHEMBL7299678

CC(C)(C)OC(=O)N=C(NC(=O)OC(C)(C)C)N1CCC(CN)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
TSHR P16473 1/20 0.36
ACACB O00763 1/20 0.36
ACACA Q13085 1/20 0.36
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
TPSAB1 Q15661 2/20 0.34
TPSD1 Q9BZJ3 2/20 0.34
TPSG1 Q9NRR2 2/20 0.34
EPHX1 P07099 1/20 0.33
ITGB3 P05106 1/20 0.32
ITGA2B P08514 1/20 0.32
DRD2 P14416 2/20 0.32
CYP2C9 P11712 1/20 0.32
HSD11B1 P28845 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CHRM2 P08172 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9073870 1.00 ALDH1A1 (0.36) ALDH1A1KMT2AMEN1TSHRACACB
SCHEMBL17574380 1.00 ALDH1A1 (0.36) ALDH1A1KMT2AMEN1TSHRACACB
SCHEMBL17574398 0.91 ACACB (0.36) ALDH1A1KMT2AMEN1TSHRACACB
SCHEMBL28173828 0.91 ACACB (0.36) ALDH1A1KMT2AMEN1TSHRACACB
SCHEMBL19410256 0.90 ACACB (0.38) ALDH1A1KMT2AMEN1TSHRACACB
SCHEMBL15080558 0.88 ALDH1A1 (0.36) ALDH1A1KMT2AMEN1TSHRACACB
SCHEMBL13519732 0.88 ALDH1A1 (0.36) ALDH1A1KMT2AMEN1TSHRACACB
SCHEMBL17574400 0.86 MEN1 (0.36) ALDH1A1KMT2AMEN1TSHRKDM4E
SCHEMBL28403064 0.86 MEN1 (0.36) ALDH1A1KMT2AMEN1TSHRKDM4E
SCHEMBL9214872 0.85 KDM4E (0.36) ALDH1A1KMT2AMEN1TSHRACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074821-B Diamide macrocycles as FXIA inhibitors 百时美施贵宝公司 2020-05-22 CN disclosed
US-5583146-A Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0648780-A1 Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1995-04-19 EP disclosed