SCHEMBL7299751

SCHEMBL7299751

O=Cc1cccc2nc(-c3ccccc3)sc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
LMNA P02545 4/20 0.44
NFKB1 P19838 3/20 0.44
NFKB2 Q00653 3/20 0.44
RELA Q04206 3/20 0.44
ALDH1A1 P00352 5/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
MAPT P10636 3/20 0.43
GLA P06280 3/20 0.43
GAA P10253 3/20 0.43
HPGD P15428 2/20 0.43
PKM P14618 1/20 0.43
APP P05067 2/20 0.42
CYP2A6 P11509 1/20 0.41
MAOB P27338 2/20 0.41
RAB9A P51151 4/20 0.39
NPC1 O15118 3/20 0.39
TP53 P04637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12649170 0.75 ALDH1A1 (0.45) KDM4ESMN1; SMN2LMNAALDH1A1MEN1
SCHEMBL543240 0.75 CYP2A6 (0.44) KDM4ESMN1; SMN2LMNAALDH1A1MEN1
SCHEMBL27925517 0.75 APP (0.45) KDM4ESMN1; SMN2LMNANFKB1NFKB2
SCHEMBL23462851 0.75 CYP2A6 (0.44) KDM4ESMN1; SMN2LMNAALDH1A1MEN1
SCHEMBL30903623 0.75 APP (0.45) KDM4ESMN1; SMN2LMNANFKB1NFKB2
SCHEMBL23462968 0.75 CYP2A6 (0.44) LMNAALDH1A1MEN1KMT2AGAA
SCHEMBL2138067 0.75 APP (0.49) KDM4ESMN1; SMN2LMNANFKB1NFKB2
SCHEMBL30594904 0.74 APP (0.49) KDM4ESMN1; SMN2LMNANFKB1NFKB2
SCHEMBL28598741 0.74 APP (0.49) KDM4ESMN1; SMN2LMNANFKB1NFKB2
SCHEMBL5116616 0.74 SMN1; SMN2 (0.51) KDM4ESMN1; SMN2LMNANFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5412099-A Intermediate benzothiazolyl- and benzoxazolyl-aldehyde compounds BAYER AKTIENGESELLSCHAFT (DE) 1995-05-02 US disclosed
EP-0450420-B1 Dihydropyridines substituted by heterocycles, process for their preparation and their use in medicaments BAYER AG (DE) 1994-09-21 EP disclosed
US-5254692-A Inotropic BAYER AKTIENGESELLSCHAFT (DE) 1993-10-19 US disclosed
US-5200420-A Inotropic agents for cardiovascular disorders BAYER AKTIENGESELLSCHAFT (DE) 1993-04-06 US disclosed
EP-0450420-A2 Dihydropyridines substituted by heterocycles, process for their preparation and their use in medicaments BAYER AG (DE) 1991-10-09 EP disclosed