SCHEMBL7300089

SCHEMBL7300089

COC(=O)[C@H](Cc1ccc(OC)cc1)NC(=O)N1C[C@@H](O)[C@@H](O)C1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.55
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
POLB P06746 1/20 0.52
GFER P55789 1/20 0.52
KDM4E B2RXH2 1/20 0.47
KMT2A Q03164 3/20 0.46
ATM Q13315 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
YAP1 P46937 3/20 0.45
NPSR1 Q6W5P4 1/20 0.45
LDHA P00338 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7295919 0.90 KMT2A (0.57) GAAPOLBKMT2ALDHATSHR
SCHEMBL7278749 0.83 CYP3A4 (0.61) GAACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7300404 0.82 POLB (0.60) GAACYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL16879017 0.77 LDHA (0.54) GAACYP2C9CYP2C19POLBKMT2A
SCHEMBL5706152 0.77 ACACB (0.58) GAACYP2C9CYP2C19KMT2AATM
SCHEMBL16879018 0.77 LDHA (0.54) GAACYP2C9CYP2C19POLBKMT2A
SCHEMBL6662892 0.77 ACACB (0.58) GAACYP2C9CYP2C19KMT2AATM
SCHEMBL8645164 0.74 LDHA (0.57) KMT2ALDHA
SCHEMBL13033619 0.74 LDHA (0.57) KMT2ALDHA
SCHEMBL9832460 0.74 LDHA (0.50) GAACYP2C9CYP2C19KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032577-A Hypotensive ABBOTT LABORATORIES (US) 1991-07-16 US disclosed
EP-0416393-A1 Peptidyl difluorodiol renin inhibitors ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
EP-0341602-A2 Renin-inhibiting functionalized peptidyl aminodiols and - triols ABBOTT LABORATORIES (US) 1989-11-15 EP disclosed