SCHEMBL7300091

SCHEMBL7300091

CN1C2COCC1CC(NC(=O)c1nn(C)c3ccccc13)C2

nearest known ligand 0.83

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.83
CYP3A4 P08684 1/20 0.83
TSHR P16473 1/20 0.83
MAPK1 P28482 1/20 0.83
HSD17B10 Q99714 1/20 0.83
HTR3A P46098 12/20 0.79
HTR3E A5X5Y0 1/20 0.79
SLC22A2 O15244 1/20 0.79
HTR3B O95264 1/20 0.79
CHRNB2 P17787 1/20 0.79
CHRNA3 P32297 1/20 0.79
CHRNA4 P43681 1/20 0.79
KCNH2 Q12809 1/20 0.79
HTR3D Q70Z44 1/20 0.79
HTR3C Q8WXA8 1/20 0.79
SLC47A1 Q96FL8 1/20 0.79
KDM4E B2RXH2 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8714556 1.00 ALDH1A1 (0.83) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL9485783 0.91 ALDH1A1 (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL30596797 0.91 ALDH1A1 (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL13660190 0.88 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL445223 0.88 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL7428799 0.88 ALDH1A1 (0.83) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL34178 0.88 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL4890 0.88 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
SCHEMBL7439648 0.88 ALDH1A1 (0.83) ALDH1A1CYP3A4TSHRMAPK1HSD17B10
Granisetron SCHEMBL4109977 0.88 HTR3A (1.00) ALDH1A1CYP3A4TSHRMAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0377967-A2 9-Aza-3-(oxa/thia)-bicyclo[3,2,1]nonane derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1990-07-18 EP claimed
EP-0708105-B1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO (JP) 1998-12-23 EP disclosed
EP-0708105-A1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1996-04-24 EP disclosed
EP-0377967-A2 9-Aza-3-(oxa/thia)-bicyclo[3,2,1]nonane derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1990-07-18 EP disclosed