SCHEMBL7300253

SCHEMBL7300253

O=C(N[C@H]1c2ccccc2C[C@@H]1O)C(Cc1ccccc1)CC(O)CC(Cc1ccccc1)C(=O)N[C@H]1c2ccccc2C[C@@H]1O

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
VIPR2 P41587 18/20 0.70
MMP9 P14780 2/20 0.64
MMP1 P03956 1/20 0.62
MMP2 P08253 1/20 0.62
MMP8 P22894 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300250 1.00 VIPR2 (0.70) VIPR2MMP9MMP1MMP2MMP8
SCHEMBL6466122 0.97 VIPR2 (0.69) VIPR2MMP9MMP1MMP2MMP8
SCHEMBL15713420 0.93 VIPR2 (0.66) VIPR2MMP9
SCHEMBL15714613 0.93 VIPR2 (0.66) VIPR2MMP9
SCHEMBL7293187 0.92 MMP9 (0.74) VIPR2MMP9MMP1MMP2MMP8
SCHEMBL7293189 0.92 MMP9 (0.74) VIPR2MMP9MMP1MMP2MMP8
SCHEMBL15713978 0.92 VIPR2 (0.64) VIPR2MMP9
SCHEMBL15713701 0.91 VIPR2 (0.65) VIPR2MMP9
SCHEMBL6468083 0.90 VIPR2 (0.62) VIPR2MMP9MMP2
SCHEMBL6469322 0.90 VIPR2 (0.64) VIPR2MMP9MMP1MMP2MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0480714-A2 HIV protease inhibitors having symmetrical structure MERCK & CO. INC. (US) 1992-04-15 EP claimed
JP-5148205-A None JP disclosed
JP-H05148205-A HIV PROTEASE INHIBITOR HAVING SYMMETRICAL STRUCTURE MERCK & CO INC 1993-06-15 JP disclosed
EP-0480714-A2 HIV protease inhibitors having symmetrical structure MERCK & CO. INC. (US) 1992-04-15 EP disclosed