SCHEMBL7300314

SCHEMBL7300314

[O]c1cc(F)c(F)c2c(F)cccc12

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.33
CES1 P23141 2/20 0.33
BCHE P06276 1/20 0.33
AR P10275 4/20 0.32
NPC1 O15118 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PGR P06401 1/20 0.31
AHR P35869 2/20 0.31
PARP1 P09874 2/20 0.31
DAO P14920 1/20 0.30
DDO Q99489 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20356033 0.80 CYP1A2 (0.35) CES2CES1BCHEARPGR
SCHEMBL13755386 0.75 CYP1A2 (0.36)
SCHEMBL5250290 0.75 ACHE (0.39) HPGDSMN1; SMN2PARP1
SCHEMBL5250287 0.75 CYP1A2 (0.33)
SCHEMBL20356032 0.71 CYP1A2 (0.35) CES2CES1BCHEARPGR
SCHEMBL7306395 0.71 CES2 (0.33) CES2CES1
SCHEMBL7305545 0.70 CES2 (0.34) CES2CES1BCHEARNPC1
SCHEMBL7305440 0.68 CYP1A2 (0.33) CES2CES1BCHEARNPC1
SCHEMBL7716701 0.67 CYP1A2 (0.39) CES2CES1BCHENPC1AHR
SCHEMBL15352162 0.66 CES2 (0.39) CES2CES1BCHENPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed