SCHEMBL7300324

SCHEMBL7300324

CC1(C)C[C]c2ccc(C#N)cc2O1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 10/20 0.37
MALT1 Q9UDY8 1/20 0.36
MAOB P27338 1/20 0.35
ABCC9 O60706 4/20 0.34
DAO P14920 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ABCC8 Q09428 2/20 0.32
KCNJ11 Q14654 2/20 0.32
KCNJ8 Q15842 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7292953 0.88 KDM4E (0.38) ABCB1MALT1MAOBABCC9KDM4E
SCHEMBL7297213 0.81 KCNE1 (0.34) ABCB1KDM4ECYP1A2CYP2D6CYP2C19
SCHEMBL7290029 0.76 AKR1B1 (0.37) MALT1MAOBCYP2D6
SCHEMBL7298546 0.76 AHR (0.35) MAOB
SCHEMBL9583441 0.73 KDM4E (0.37) ABCB1MALT1KDM4E
SCHEMBL25387439 0.71 DAO (0.41) ABCB1MALT1MAOBABCC9DAO
SCHEMBL30514069 0.71 DAO (0.41) ABCB1MALT1MAOBABCC9DAO
SCHEMBL7299826 0.71 AKR1B1 (0.42) MALT1
SCHEMBL7300321 0.70 ABCB1 (0.38) ABCB1MALT1MAOBABCC9DAO
SCHEMBL7292321 0.69 PKM (0.35) ABCB1MAOBDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260444-A Cardiovascular, hypotensive WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed
US-5208245-A Hypotensive agents WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-05-04 US disclosed
EP-0460418-A2 Novel Dihydropyridine derivative WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1991-12-11 EP disclosed