SCHEMBL7300700

SCHEMBL7300700

CCCCN(C(=O)NC1CCCCC1)c1cc(C)c2nc(CCC)n(Cc3ccc(-c4ccccc4-c4nnn[nH]4)cc3)c2c1

nearest known ligand 0.53

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 15/20 0.46
AGTR2 P50052 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308640 0.94 AGTR1 (0.47) AGTR1AGTR2
SCHEMBL7309365 0.91 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL8873636 0.88 AGTR1 (0.44) AGTR1AGTR2
SCHEMBL7303448 0.88 AGTR1 (0.60) AGTR1AGTR2
SCHEMBL7303454 0.86 AGTR1 (0.48) AGTR1AGTR2
Water SCHEMBL8789674 0.85 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL8789331 0.85 AGTR1 (0.55) AGTR1AGTR2
SCHEMBL7303128 0.85 AGTR1 (0.55) AGTR1AGTR2
Water SCHEMBL8789127 0.85 AGTR1 (0.55) AGTR1AGTR2
SCHEMBL7302489 0.84 AGTR1 (0.48) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614519-A (1-(2,3 or 4-N-morpholinoalkyl)-imidazol-4-yl)-benizimidazol-1-yl-methyl]-biphenyls useful as angiotensin-II antagonists KARL THOMAE GMBH (DE) 1997-03-25 US disclosed
US-5602127-A ADMINISTERING TO TREAT HYPERTENSION KARL THOMAE GMBH (DE) 1997-02-11 US disclosed
US-5594003-A HYPOTENSIVE AGENTS DR. KARL THOMAE GMBH (DE) 1997-01-14 US disclosed
US-5591762-A HYPOTENSIVE AGENTS DR. KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
EP-0502314-A1 Benzimidazol, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-09 EP disclosed