SCHEMBL7301080

SCHEMBL7301080

CC1(C)C[CH]c2cc(OC(F)(F)F)ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
SLC6A4 P31645 3/20 0.35
GPR3 P46089 2/20 0.35
P2RY1 P47900 1/20 0.35
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
BACE1 P56817 2/20 0.34
CTSD P07339 1/20 0.34
SLC6A3 Q01959 2/20 0.34
TRPV1 Q8NER1 3/20 0.34
CYP2D6 P10635 2/20 0.34
CYP3A4 P08684 1/20 0.34
CES1 P23141 1/20 0.33
ABL1 P00519 1/20 0.33
PPARA Q07869 3/20 0.32
PPARD Q03181 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7291317 0.88 TRPV1 (0.36) PTGS1PTGS2SLC6A4GPR3P2RY1
SCHEMBL9584799 0.81 CA12 (0.40) CA12CA9BACE1CTSDCYP3A4
SCHEMBL7300076 0.77 PTGS1 (0.35) PTGS1PTGS2CA12CA9BACE1
SCHEMBL8802196 0.75 HIF1A (0.43) PTGS1PTGS2CA12CA9CYP3A4
SCHEMBL7294955 0.74 HTR2C (0.42)
SCHEMBL7301082 0.72 P2RY1 (0.36) PTGS1PTGS2SLC6A4GPR3P2RY1
SCHEMBL7294557 0.71 HTR2C (0.42) CA12CA9BACE1CTSD
SCHEMBL2350567 0.71 BACE1 (0.36) CA12CA9BACE1CTSD
SCHEMBL7134096 0.71 MAPT (0.49) PTGS1PTGS2CA12CA9CYP3A4
SCHEMBL7293216 0.71 PTGS1 (0.41) PTGS1PTGS2GPR3CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260444-A Cardiovascular, hypotensive WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed
US-5208245-A Hypotensive agents WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-05-04 US disclosed
EP-0460418-A2 Novel Dihydropyridine derivative WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1991-12-11 EP disclosed