SCHEMBL7301113

SCHEMBL7301113

CC(C)(C)OC(=O)NC(CC(=O)C(Cc1ccccc1)NC(=O)OC(C)(C)C)Cc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACE P12821 3/20 0.65
ATM Q13315 1/20 0.64
CTSS P25774 6/20 0.61
CTSK P43235 5/20 0.61
CTSB P07858 2/20 0.61
CTSL P07711 1/20 0.61
APP P05067 3/20 0.58
CA2 P00918 1/20 0.55
KLK5 Q9Y337 1/20 0.55
AKT1 P31749 1/20 0.54
REN P00797 1/20 0.52
PPARA Q07869 2/20 0.51
PPARG P37231 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL489490 0.87 ATM (0.70) ACEATMCTSSCTSKCTSB
SCHEMBL489489 0.87 ATM (0.70) ACEATMCTSSCTSKCTSB
SCHEMBL1519945 0.87 ATM (0.70) ACEATMCTSSCTSKCTSB
SCHEMBL7324443 0.86 ACE (0.67) ACEATMCTSSCTSKCTSB
SCHEMBL10376903 0.86 ACE (0.67) ACEATMCTSSCTSKCTSB
SCHEMBL7329244 0.86 ACE (0.67) ACEATMCTSSCTSKCTSB
SCHEMBL21834807 0.86 ATM (0.65) ACEATMCTSSCTSKCTSB
SCHEMBL6516027 0.85 ACE (0.70) ACEATMCTSSCTSKCTSB
SCHEMBL17688687 0.85 ACE (0.70) ACEATMCTSSCTSKCTSB
SCHEMBL2603668 0.85 ACE (0.70) ACEATMCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed