SCHEMBL7301685

SCHEMBL7301685

CCCC(CC[C]=O)N1CCCC1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 18/20 0.35
SLC6A2 P23975 15/20 0.35
SLC6A4 P31645 11/20 0.34
HRH3 Q9Y5N1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL898138 0.83 SLC6A3 (0.39) SLC6A3SLC6A2SLC6A4HRH3
Iodide SCHEMBL15008876 0.81 SLC6A3 (0.38) SLC6A3SLC6A2SLC6A4HRH3
SCHEMBL3302667 0.81 SLC6A3 (0.38) SLC6A3SLC6A2SLC6A4HRH3
SCHEMBL13182550 0.81 SLC6A3 (0.32) SLC6A3SLC6A2SLC6A4
SCHEMBL22701318 0.79 SLC6A3 (0.35) SLC6A3SLC6A2SLC6A4HRH3
SCHEMBL14160126 0.75 HRH3 (0.40) SLC6A3SLC6A2SLC6A4HRH3
SCHEMBL2229569 0.74 SLC6A3 (0.37) SLC6A3SLC6A2SLC6A4
SCHEMBL24869964 0.74 HRH3 (0.42) SLC6A3SLC6A2SLC6A4HRH3
SCHEMBL18403963 0.74 SLC6A3 (0.34) SLC6A3SLC6A2SLC6A4HRH3
SCHEMBL14204509 0.74 HRH3 (0.42) SLC6A3SLC6A2SLC6A4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378691-A Amino acid derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-01-03 US disclosed
EP-0501280-A2 Renin-inhibiting peptide analogues MERCK PATENT GmbH (DE) 1992-09-02 EP disclosed
EP-0446485-A2 Peptide analogues with renininhibiting activity MERCK PATENT GmbH (DE) 1991-09-18 EP disclosed
EP-0418696-A2 Derivatives of aminoacids MERCK PATENT GmbH (DE) 1991-03-27 EP disclosed
EP-0339483-A2 Renin inhbiting amino-acid derivatives MERCK PATENT GmbH (DE) 1989-11-02 EP disclosed