SCHEMBL7302009

SCHEMBL7302009

COc1ccc2c(c1)CCC(CC(=O)C1C(=S)CN[C@@H]1C(=O)O)C2

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 1/20 0.47
CYP19A1 P11511 2/20 0.44
SIGMAR1 Q99720 2/20 0.42
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
ACHE P22303 2/20 0.41
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
MCHR1 Q99705 2/20 0.38
HTR1A P08908 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294598 0.89 CYP26A1 (0.44) CYP26A1CYP19A1SIGMAR1CA1CA2
SCHEMBL7295069 0.87 CYP26A1 (0.42) CYP26A1CYP19A1SIGMAR1CA1CA2
SCHEMBL7301359 0.86 ITGB3 (0.37) CYP26A1ITGB3ITGA2BMCHR1
SCHEMBL7294732 0.85 DPP4 (0.44) CYP26A1CYP19A1SIGMAR1CA1CA2
SCHEMBL7301552 0.84 PREP (0.39) CYP19A1SIGMAR1ADRA1DADRA1AADRA1B
SCHEMBL7295266 0.84 PREP (0.39) CYP19A1SIGMAR1ADRA1DADRA1AADRA1B
SCHEMBL7294861 0.84 PREP (0.39) CYP19A1SIGMAR1ADRA1DADRA1AADRA1B
SCHEMBL7296404 0.78 GAA (0.36)
SCHEMBL4621033 0.78 CYP26A1 (0.61) CYP26A1CYP19A1SIGMAR1CA1CA2
SCHEMBL7297223 0.77 ITGB3 (0.34) CYP26A1ITGB3ITGA2BDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017929-A Cholinesterase activator ZERIA PHARMACEUTICAL CO., LTD. (JP) 2000-01-25 US disclosed
EP-0754454-A1 CHOLINESTERASE ACTIVATOR ZERIA PHARMACEUTICAL CO., LTD. (JP) 1997-01-22 EP disclosed
EP-0372484-B1 Condensed benzene derivative ZERIA PHARM CO LTD (JP) 1994-10-26 EP disclosed
US-5028604-A Cognition Activators ZERIA PHARMACEUTICAL CO., LTD. (JP) 1991-07-02 US disclosed
EP-0372484-A2 Condensed benzene derivative ZERIA PHARMACEUTICAL CO., LTD. (JP) 1990-06-13 EP disclosed