SCHEMBL7302500

SCHEMBL7302500

[NH]C(=O)/C=C(\C(=O)O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 3/20 0.55
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
KMT2A Q03164 4/20 0.46
NFE2L2 Q16236 1/20 0.43
AKR1C2 P52895 2/20 0.43
AKR1C3 P42330 1/20 0.43
ALDH1A1 P00352 4/20 0.42
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
TSHR P16473 2/20 0.42
DAO P14920 1/20 0.42
NAPRT Q6XQN6 1/20 0.42
PTGS2 P35354 1/20 0.42
TDP1 Q9NUW8 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPK1 P28482 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL164579 0.82 AKR1C1 (0.59) AKR1C1CA12CA1CA2CA9
SCHEMBL165294 0.82 AKR1C1 (0.59) AKR1C1CA12CA1CA2CA9
SCHEMBL164580 0.82 AKR1C1 (0.59) AKR1C1CA12CA1CA2CA9
SCHEMBL27489619 0.80 NFE2L2 (0.61) AKR1C1CA12CA1CA2CA9
SCHEMBL4793306 0.80 CA12 (0.65) AKR1C1CA12CA1CA2CA9
Hydrochloric Acid SCHEMBL3674640 0.80 AKR1C1 (0.57) AKR1C1CA12CA1CA2CA9
SCHEMBL4730610 0.80 NFE2L2 (0.61) AKR1C1CA12CA1CA2CA9
SCHEMBL9248787 0.78 AKR1C1 (0.55) AKR1C1CA12CA1CA2CA9
SCHEMBL8440602 0.78 AKR1C1 (0.55) AKR1C1CA12CA1CA2CA9
SCHEMBL5273972 0.78 AKR1C1 (0.55) AKR1C1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0468470-B1 Benzimidazoles, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1997-04-16 EP disclosed
EP-0502314-A1 Benzimidazol, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-09 EP disclosed
EP-0468470-A1 Benzimidazoles, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-01-29 EP disclosed